Jaime Escalante García
Doctorado en Química Orgánica, CINVESTAV-IPN (1995)
Profesor: Titular C
SNI: Nivel II
Líneas de Investigación:
Laboratorio de Sintésis Asimétrica
Cuerpo Académico: Química Farmacéutica y Biotecnología
jaime@uaem.mx |Teléfono: +52 777 329 79 97 Ext. 6040
ORCID: 0000-0001-5485-0244| Scopus Author ID: 7003360738|
2024
78. Flores-Hernández, F., Zárate-López, T. I., Alcaráz-Cano, M. A., Escalante, J., & Rivera-Ramírez, J. D. (2024). Podophyllotoxin and Aryltetralin Lignans: Methods for the Synthesis of Rings A, B, C, D. Journal of Organic and Pharmaceutical Chemistry, 22(2), 3–25. https://doi.org/10.24959/ophcj.24.308942
77. Chavelas-Hernández, Leticia y Hernández-Vázquez, Luis G. y Valdez-Camacho, Jonathan R. y Espinoza-Guillén, Adrián y Tavira-Montalván, Carlos A. y Meneses-Acosta, Angélica y Juaristi, Eusebio y Ruiz-Azuara, Lena y Escalante, Jaime, Síntesis de complejos de nitrato de cobre (1,10-fenantrolina- K 2 N ,N')(Β 2 -metil- y Β 2 -fenilalaninato- K 2 N ,O) y su actividad antiproliferativa en las líneas celulares de cáncer Mcf-7 y A549. Disponible en SSRN: https://ssrn.com/abstract=4758164 o http://dx.doi.org/10.2139/ssrn.4758164
75. Bahena‐Martínez, J. D., Flores, R., Domínguez‐Mendoza, B. E., Hernández‐Vázquez, L. G., Juaristi, E., & Escalante, J*. (2024). Synthesis of β‐Truxinate via [2+2] Cycloaddition of Methyl 4‐Nitrocinnamate: Kinetic Study of its Isomerization with DBU. ChemistrySelect, 9(22). https://doi.org/10.1002/slct.202400178
2023
74. Guzmán-Ávila, R., Estrada-Soto, S*., Arias-Durán, L., Millán-Pacheco, C., Escalante-García, J., Rios, M. Y., Flores-Morales, V., Villalobos-Molina, R., & Pérez-Barrón, G. (2023). Vasorelaxant and Antihypertensive Effects of (3β)-ursen-12-en-3,28-diol by NO/cGMP System. Letters in Drug Design & Discovery, 20(12), 1959–1969. DOI: 10.2174/1570180819666220704111424
73. Chavelas-Hernández, L., Hernández-Vázquez, L. G., Bahena-Martínez, J. D., Arroyo-Colín, A. B., Flores-Osorio, S. G., Navarrete-Vázquez, G., & Escalante, J. (2023). Aza-Michael Additions of Benzylamine to Acrylates Promoted by Microwaves and Conventional Heating Using DBU as Catalyst via Solvent-Free Protocol. Processes, 12(1), 34. DOI: 10.3390/pr12010034
72. Romero-Ibañez, J., Ortega-Rojas, M. A., Valdéz-Camacho, J. R., Hernández-Vázquez, L. G., Sartillo-Piscil, F., & Escalante, J.* (2023). Asymmetric Synthesis of trans-3-Alkoxyamino-4-Oxygenated-2-Piperidones Mediated by Transition-Metal-Free Dual C-H Oxidation and Its CAL-B-Assisted Enzymatic Resolution. Catalysts, 13(4), 703. DOI: 10.3390/catal13040703
2022
71. Sánchez‐Muñoz, G. K.; Ortega‐Rojas, M. A*.; Chavelas‐Hernández, L.; Razo‐Hernández, R. S.; Valdéz‐Camacho, J. R.; Escalante, J*. Solvent‐Free Lipase‐Catalyzed Transesterification of Alcohols with Methyl Esters Under Vacuum‐Assisted Conditions. ChemistrySelect 2022, 7 (30). DOI: 10.1002/slct.202202643.
2021
70. Ortega‐Rojas, M. A.; Castillo, E*.; Razo‐Hernández, R. S.; Pastor, N.; Juaristi, E.; Escalante, J.* Effect of the Substituent and Amino Group Position on the Lipase‐Catalyzed Resolution of γ‐Amino Esters: A Molecular Docking Study Shedding Light on Candida Antarctica Lipase B Enantioselectivity. European J. Org. Chem. 2021, 2021 (34), 4790–4802. DOI: 10.1002/ejoc.202100712
2020
69. Méndez, A.; Valdez-Camacho, J. R.; Escalante, J.* Photooxidation of 2-(Tert-Butyl)-3-Methyl-2,3,5,6,7,8-Hexahydroquinazolin-4(1H)-One, an Example of Singlet Oxygen Ene Reaction. Molecules 2020, 25 (21), 5008 DOI: 10.3390/molecules25215008
68. Valdéz-Camacho, J. R., Ramírez-Solís, A., Escalante, J., Ruiz-Azuara, L., & Hô, M.* (2020). Theoretical determination of half-wave potentials for phenanthroline-, bipyridine-, acetylacetonate-, and glycinate-containing copper (II) complexes. Journal of Molecular Modeling, 26(7), 191. https://doi.org/10.1007/s00894-020-04453-x
ARTÍCULOS EN REVISTAS INDEXADAS
2023
72. Romero-Ibañez, J., Ortega-Rojas, M. A., Valdéz-Camacho, J. R., Hernández-Vázquez, L. G., Sartillo-Piscil, F., & Escalante, J.* (2023). Asymmetric Synthesis of trans-3-Alkoxyamino-4-Oxygenated-2-Piperidones Mediated by Transition-Metal-Free Dual C-H Oxidation and Its CAL-B-Assisted Enzymatic Resolution. Catalysts, 13(4), 703. DOI: 10.3390/catal13040703
2022
71. Sánchez‐Muñoz, G. K.; Ortega‐Rojas, M. A*.; Chavelas‐Hernández, L.; Razo‐Hernández, R. S.; Valdéz‐Camacho, J. R.; Escalante, J*. Solvent‐Free Lipase‐Catalyzed Transesterification of Alcohols with Methyl Esters Under Vacuum‐Assisted Conditions. ChemistrySelect 2022, 7 (30). DOI: 10.1002/slct.202202643.
2021
70. Ortega‐Rojas, M. A.; Castillo, E*.; Razo‐Hernández, R. S.; Pastor, N.; Juaristi, E.; Escalante, J.* Effect of the Substituent and Amino Group Position on the Lipase‐Catalyzed Resolution of γ‐Amino Esters: A Molecular Docking Study Shedding Light on Candida Antarctica Lipase B Enantioselectivity. European J. Org. Chem. 2021, 2021 (34), 4790–4802. DOI: 10.1002/ejoc.202100712
2020
69. Méndez, A.; Valdez-Camacho, J. R.; Escalante, J.* Photooxidation of 2-(Tert-Butyl)-3-Methyl-2,3,5,6,7,8-Hexahydroquinazolin-4(1H)-One, an Example of Singlet Oxygen Ene Reaction. Molecules 2020, 25 (21), 5008 DOI: 10.3390/molecules25215008
68. Valdéz-Camacho, J. R., Ramírez-Solís, A., Escalante, J., Ruiz-Azuara, L., & Hô, M.* (2020). Theoretical determination of half-wave potentials for phenanthroline-, bipyridine-, acetylacetonate-, and glycinate-containing copper (II) complexes. Journal of Molecular Modeling, 26(7), 191. https://doi.org/10.1007/s00894-020-04453-x
67. Valdez-Camacho, J. R.; Pérez-Salgado, Y.; Espinoza-Guillén, A.; Gómez-Vidales, V.; Alberto Tavira-Montalvan, C.; Meneses-Acosta, A.; Leyva, M. A.; Vázquez-Ríos, M. G.; Juaristi, E.; Höpfl, H.; Ruiz-Azuara, L.; Escalante, J.* Synthesis, Structural Characterization and Antiproliferative Activity on MCF-7 and A549 Tumor Cell Lines of [Cu(N-N)(Β3-Aminoacidate)]NO3 Complexes (Casiopeínas®). Inorganica Chim. Acta 2020, 506, 119542 DOI: 10.1016/j.ica.2020.119542
2019
66. Chavelas-Hernández, L.; Valdéz-Camacho, J. R.; Hernández-Vázquez, L. G.; Dominguez-Mendoza, B. E.; Vasquez-Ríos, M. G.; Escalante, J.* A New Approach Using Aromatic-Solvent-Induced Shifts in NMR Spectroscopy to Analyze β-Lactams with Various Substitution Patterns. Synlett 2019 DOI: 10.1055/s-0039-1691498
65. Álvarez-Santamaría, L.; Juaristi, E.; Arroyo-Colín, A. B.; Palma-Flores, J.; Cabrera-Rivera, F. A.; Escalante, J.* Efficient Solvent-Free Preparation of Imines, and Their Subsequent Oxidation with ≪I≫M≪/I≫-CPBA to Afford Oxaziridines. Green Sustain. Chem. 2019, 09 (04), 143–154 DOI: 10.4236/gsc.2019.94011
64. Valdez‐Camacho, J. R.; Cortés‐Guzmán, K. P.; Torres‐Gómez, H.; Flores, R.; Leyva, M. A.; Escalante, J.* Kinetics, Thermodynamics, and Theoretical Studies in a Diels‐Alder Dimerization Process of 3‐Vinylindole Derivative of the 3‐Indoleacetic Acid: An Auxin. ChemistrySelect 2019, 4 (28), 8311–8316. DOI: 10.1002/slct.201901141
63. Morales-Vilchis, M. G.; Flores-Sánchez, P.; Escalante, J. Identification, Synthesis and Structure Assignment of Two Impurities of Erlotinib, a Drug Used for the Treatment of Some Types of Cancer. J. Mex. Chem. Soc. 2019, 63 (1) DOI: 10.29356/jmcs.v63i1.714
62. Valdéz-Camacho, J. R.; Rivera-Ramírez, J. D.; Escalante, J.* Studies and Mechanism of Olefination Reaction in Aryl-Enolates with Paraformaldehyde. Int. J. Org. Chem. 2019, 09 (01), 10–22. DOI: 10.4236/ijoc.2019.91002
2017
61. Cabrera-Rivera, F. A.; Hernández-Vázquez, L. G.; Flores-Sánchez, P.; Durán-Galván, M.; Escalante, J.* Solvent- and Catalyst-Free Microwave-Assisted Decarboxylation of Malonic Acid Derivatives. Green Sustain. Chem. 2017, 7 (4), 270–280. DOI: 10.4236/gsc.2017.74021
60. Ortega-Rojas, M.; Rivera-Ramírez, J.; Ávila-Ortiz, C.; Juaristi, E.*; González-Muñoz, F.; Castillo, E.*; Escalante, J.* One-Pot Lipase-Catalyzed Enantioselective Synthesis of (R)-(−)-N-Benzyl-3-(Benzylamino)butanamide: The Effect of Solvent Polarity on Enantioselectivity. Molecules 2017, 22 (12), 2189. DOI: 10.3390/molecules22122189
59. Pérez-Venegas, M.; Reyes-Rangel, G.; Neri, A.; Escalante, J.*; Juaristi, E.* Mechanochemical Enzymatic Resolution of N -Benzylated-β 3 -Amino Esters. Beilstein J. Org. Chem. 2017, 13, 1728–1734. DOI: 10.3762/bjoc.13.167
2016
58. Torres-Huerta, A.; Cruz-Huerta, J.; Höpfl, H.*; Hernández-Vázquez, L. G.; Escalante-García, J.; Jiménez-Sánchez, A.; Santillan, R.; Hernández-Ahuactzi, I. F.; Sánchez, M. Variation of the Molecular Conformation, Shape, and Cavity Size in Dinuclear Metalla-Macrocycles Containing Hetero-Ditopic Dithiocarbamate–Carboxylate Ligands from a Homologous Series of N-Substituted Amino Acids. Inorg. Chem. 2016. DOI: 10.1021/acs.inorgchem.6b02387
57. Rosas-Valdéz, M. E.; Escalante, J.*; Bustos-Jaimes, I.; Regla, I.; Boto, A. Synthesis and Modification of the Amyloid Peptide Sequence 37-42 of Aβ42 (AβPP): Efficient Synthesis of N-Methylated Peptides, Expanding the Tools for Peptide Research. J. Mex. Chem. Soc. 2016, 60 (3), 125–134. Online
56. Boto, A.; Escalante, J. 1‐(Trimethylsilyl)‐1H‐benzotriazole. e-EROS Encycl. Reagents Org. Synth. DOI: 10.1002/047084289X.rn01189
2015
55. Rangel, H.; Carrillo-Morales, M.; Galindo, J. M.; Castillo, E.; Obregón-Zúñiga, A.; Juaristi, E.; Escalante, J.* Structural Features of N-Benzylated-β-Amino Acid Methyl Esters Essential for Enantiodifferentiation by Lipase B from Candida Antarctica in Hydrolytic Reactions. Tetrahedron: Asymmetry 2015, 26 (7), 325–332. DOI: 10.1016/j.tetasy.2015.02.007
54. Rivera-Ramírez, J. D.; Escalante, J.*; López-Munguía, A.; Marty, A.; Castillo, E.* Thermodynamically Controlled Chemoselectivity in Lipase-Catalyzed Aza-Michael Additions. J. Mol. Catal. B Enzym. 2015, 112, 76–82. DOI: 10.1016/j.molcatb.2014.12.009
2014
53. Cabrera-Rivera, F. A.; Escalante, J.* Synthesis, Resolution and Absolute Configuration of 2, 3-Dihydro-2-Tert-Butyl-3-N-Benzylquinazolin-4-One: A Possible Chiral Auxiliary for Synthesis of β-Amino Cyclohexancarboxylic Acid. Int. J. Org. Chem. 2014, 2014. DOI: 10.4236/ijoc.2014.41007
52. Robledo, N.*; Vega, M.; Escalante, J.; Arzuffi, R. A New Component of the Male Papaya Fruit Fly (Diptera: Tephritidae) Sex Pheromone. Florida Entomol. 2014, 97 (3), 1260–1262. DOI: 10.1653/024.097.0338
51. Del-Oso, J.-A.; Maldonado, J.-L.*; Ramos-Ortíz, G*.; Rodríguez, M.; Güizado-Rodríguez, M.*; Escalante, J.; Frontana-Uribe, B. A.; Pérez-Gutiérrez, E.; Santillan, R. New Polythiophene Derivatives and Enhanced Photovoltaic Effect by a Boron Compound Blended with Them in OPVs Cells. Synth. Met. 2014, 196, 83–91. DOI: 10.1016/j.synthmet.2014.07.019
50. Cabrera-Rivera, F. A.; Escalante, J.*; Morales-Rojas, H.; Zigler, D. F.; Schmidt, R. D.; Jarocha, L. E.; Forbes, M. D. E.* Photophysical Properties of 2, 3-Dihydroquinazolin-4 (1H)-One Derivatives. J. Photochem. Photobiol. A Chem. 2014, 294, 31–37. DOI: 10.1016/j.jphotochem.2014.07.005
2012
49. Cervantes Cuevas, H.*; García Martínez, C.; Escalante García, J. Reacción de N, N’-bis (2-Heteroaril) Etilendiaminas Con Aldehídos, Nuevas Imidazolidinas. Rev. Latinoam. química 2012, 40 (3), 187–198. Online
48. Navarrete-Vazquez.*; Ramírez-Martínez, M., Estrada-Soto, S., Nava-Zuazo, C., Paoli, P., Camici, G., Escalante-García, J., (...), Ortiz-Andrade, R., G. Synthesis, in Vitro and in Silico Screening of Ethyl 2-(6-Substituted Benzo[d]thiazol-2-Ylamino)-2-Oxoacetates as Protein-Tyrosine Phosphatase 1B Inhibitors. Eur. J. Med. Chem. 2012, 53, 346–355. DOI: 10.1016/j.ejmech.2012.04.025
47. Hernández‐Vázquez, L. G.; Leyva, M. A.; Metta‐Magaña, A. J.; Escalante, J.* Microwave‐Assisted Synthesis of β‐Lactams and Cyclo‐β‐dipeptides. Helv. Chim. Acta 2012, 95 (11), 2218–2230. DOI: 10.1002/hlca.201200449
46. Cabrera-Rivera, F. A.; Ortíz-Nava, C.; Escalante, J.*; Hernández-Pérez, J. M.; Hô, M. Photoinduced Elimination in 2, 3-Dihydro-2-Tert-Butyl-3-Benzyl-4 (1H)-Quinazolinone: Theoretical Calculations and Radical Trapping Using TEMPO Derivatives. Synlett 2012, 23 (7), 1057–1063. DOI: 10.1055/s-0031-1290492
45. Sandoval-González, A.; Borja-Arco, E.; Escalante, J.; Jiménez-Sandoval, O.; Gamboa, S. A.* Methanol Oxidation Reaction on PtSnO 2 Obtained by Microwave-Assisted Chemical Reduction. Int. J. Hydrogen Energy 2012, 37 (2), 1752–1759. DOI: 10.1016/j.ijhydene.2011.10.049
44. Cabrera-Rivera, F. A.; Ortíz-Nava, C.; Román-Bravo, P.; Leyva, M. A.; Escalante, J.* Direct Halogenation Reactions in 2, 3-Dihydro-4 (1H)-Quinazolinones. Heterocycles 2012, 85 (9), 2173. DOI: 10.3987/COM-12-12473
2011
43. Borja-Arco, E.*; Jiménez-Sandoval, O.; Escalante-García, J.; Magallón-Cacho, L.; Sebastian, P. J.* Microwave Assisted Synthesis of Osmium Electrocatalysts for the Oxygen Reduction Reaction in the Absence and Presence of Aqueous Methanol. Int. J. Electrochem. 2011, 2011. DOI: 10.4061/2011/830541
42. Borja-Arco, E.; Sandoval, O. J.; Escalante-García, J.; Sandoval-González, A.; Sebastian, P. J.* Microwave Assisted Synthesis of Ruthenium Electrocatalysts for Oxygen Reduction Reaction in the Presence and Absence of Aqueous Methanol. Int. J. Hydrogen Energy 2011, 36 (1), 103–110. DOI: 10.1016/j.ijhydene.2010.10.051
41. Garcia-Martinez, C.*; Cervantes, H.; Mendez, F.; Escalante, J. Stoichiometry, Association Constant, and Solvation Model of Chiral Hydroxyfuranones in the Presence of Pirkle’s Alcohols. Spectrosc. Lett. 2011, 44 (3), 168–175. DOI: 10.1080/00387010.2010.489096
40. Nicho, M. E.*; Medrano-Baca, M. G.; León-Silva, U.; Escalante, J.; González-Rodríguez, G.; Güizado-Rodríguez, M.; Linzaga-Elizalde, I. Effect of Adhesion Promoter in Corrosion Protection of 1018 Mild Steel by Using Poly (3-Hexylthiophene) Coatings in 0.5 M H2SO4 Solution. Corros. J. Sci. Eng. 2011, 67 (10), 105002. DOI: 10.5006/1.3647763
2010
39. Güizado-Rodríguez, M.*; López-Tejeda, M.; Escalante, J.; Guerrero-Álvarez, J. A.; Nicho, M. E. Photosensitive Polyaniline Colloidal Particles Prepared by Enzymatic Polymerization Using the Azopolymer DMA-Co-AZAAm as Stabilizer. Mater. Chem. Phys. 2010, 124 (1), 389–394. DOI: 10.1016/j.matchemphys.2010.06.052
38. Miranda-Molina, A.; López-Munguía, A.; San Román, M. L.; Escalante, J.; Leyva, M. A.; Puebla, A. M.; Castillo, E.*; Álvarez, L.* Stereoselective Enzymatic Synthesis of Monoglucosyl-Myo-Inositols with in Vivo Anti-Inflammatory Activity. Tetrahedron: Asymmetry 2010, 21 (1), 43–50. DOI: 10.1016/j.tetasy.2009.12.009
2009
37. Robledo, N.; Escalante, J.*; Arzuffi, R. Extraction with SPME and Synthesis of 2-Methyl-6-Vinylpyrazine by a “One Pot”reaction Using Microwaves. Molecules 2009, 14 (6), 2160–2166. DOI: 10.3390/molecules14062160
36. Díaz-Coutiño, F. D.; Escalante, J.* Efficient ’One Pot’ Nitro Reduction-Protection of γ-Nitro Aliphatic Methyl Esters. J. Mex. Chem. Soc. 2009, 53 (3), 93–95. Online
35. Escalante, J.*; Díaz-Coutiño, F. D. Synthesis of γ-Nitro Aliphatic Methyl Esters via Michael Additions Promoted by Microwave Irradiation. Molecules 2009, 14 (4), 1595–1604. DOI: 10.3390/molecules14041595
34. Priego, J.; Ortíz-Nava, C.; Carrillo-Morales, M.; López-Munguía, A.; Escalante, J.*; Castillo, E.* Solvent Engineering: An Effective Tool to Direct Chemoselectivity in a Lipase-Catalyzed Michael Addition. Tetrahedron 2009, 65 (2), 536–539. DOI: 10.1016/j.tet.2008.10.103
33. Linzaga-Elizalde, I.*; Escalante, J.; Nicho, M. E.; Güizado-Rodríguez, M. Synthesis of 2-(Thiophen-3-Yl) Vinylphosphonic Acid. Synth. Commun. 2009, 39 (9), 1511–1515. DOI: 10.1080/00397910902784462
32. Marquina, S.; Parra, J. L.; González, M.; Zamilpa, A.; Escalante, J.; Trejo-Hernández, M. R.; Álvarez, L.* Hydroxylation of the Diterpenes Ent-Kaur-16-En-19-Oic and Ent-Beyer-15-En-19-Oic Acids by the Fungus Aspergillus Niger. Phytochemistry 2009, 70 (17), 2017–2022. DOI: 10.1016/j.phytochem.2009.09.005
31. Pérez-Picaso, L.; Escalante, J.; Olivo, H. F.; Rios, M. Y.* Efficient Microwave Assisted Syntheses of 2,5-Diketopiperazines in Aqueous Media. Molecules 2009, 14 (8), 2836–2849. DOI: 10.3390/molecules14082836
2008
30. Escalante, J. Enzymatic Resolution of β‐Amino Methyl Esters Using Lipase B from Candida Antarctica. In recent developments in physical chemistry: third mexican meeting on mathematical and experimental physics; AIP Publishing, 2008; Vol. 979, pp 60–67. DOI:10.1063/1.2901848
29. Escalante, J.*; Carrillo-Morales, M.; Linzaga, I. Michael Additions of Amines to Methyl Acrylates Promoted by Microwave Irradiation. Molecules 2008, 13 (2), 340–347. DOI: 10.3390/molecules13020340
28. Cruz-Huerta, J.; Carillo-Morales, M.; Santacruz-Juárez, E.; Hernández-Ahuactzi, I. F.; Escalante-García, J.; Godoy-Alcantar, C.; Guerrero-Alvarez, J. A.; Höpfl, H.*; Morales-Rojas, H.; Sánchez, M. Macrocyclic Diorganotin Complexes of γ-Amino Acid Dithiocarbamates as Hosts for Ion-Pair Recognition. Inorg. Chem. 2008, 47 (21), 9874–9885. DOI: 10.1021/ic8007987
2007
27. Escalante, J.*; Ortíz-Nava, C.; Flores, P.; Priego, J. M.; García-Martínez, C.* Synthesis, NMR and Crystallographic Studies of 2-Substituted Dihydroquinazolinones Derived from (S)-Phenylethylamine. Molecules 2007, 12 (2), 173–182. DOI: 10.3390/12020173
26. Torres-Gavilán, A.; Escalante, J.; Regla, I.; López-Munguía, A.; Castillo, E.* “Easy-On, Easy-Off”resolution of Chiral 1-Phenylethylamine Catalyzed by Candida Antarctica Lipase B. Tetrahedron: Asymmetry 2007, 18 (22), 2621–2624. DOI: 10.1016/j.tetasy.2007.10.045
2006
25. García-Martínez, C.*; Pérez-Espino, M. A.; Cervantes-Cuevasl, I. H.; Escalante-García, J. Synthesis of mB—Epoxysulfoxides: Thermodynamic Control in Base—induced Cyclization of Chlorohydrins Derived from a—Chlorobenzyl Phenyl Sulfoxide and Alkyl Aldehydes. 2006. Online
24. Campo, M. A.; Escalante, J.; Sebesta, R. β 2-Amino Acids with Proteinogenic Side Chains and Corresponding Peptides: Synthesis, Secondary Structure, and Biological Activity. EnantioselectiVe Synth. β-Amino Acids 2006, 593–617. DOI: 10.1002/0471698482.ch23
23. González‐Juárez, E.; Ortega‐Guevara, A.; Linzaga‐Elizalde, I.*; Escalante, J. NMR and X‐ray Crystallographic Studies of Linear and Cyclic Aminomethanephosphinates. Heteroat. Chem. 2006, 17 (2), 81–87. DOI: 10.1002/hc.20179
2005
22. Arvidsson, P. I.; Ryder, N. S.; Weiss, H. M.; Hook, D. F.; Escalante, J.; Seebach, D.* Exploring the Antibacterial and Hemolytic Activity of Shorter-and Longer-Chain B-, A, B-, and G-Peptides, and of B-Peptides from β2 -3-Aza-and b3-2-Methylidene-Amino Acids Bearing Proteinogenic Side Chains-A Survey. Chem. Biodivers. 2005, 2, 401. DOI: 10.1002/cbdv.200590020
21. Flores-Sánchez, P.; Escalante, J.*; Castillo, E. Enzymatic Resolution of N-Protected-β 3-Amino Methyl Esters, Using Lipase B from Candida Antarctica. Tetrahedron: Asymmetry 2005, 16 (3), 629–634. DOI: 10.1016/j.tetasy.2004.11.082
2004
20. Bivián-Castro, E. Y.; Bernes, S.; Escalante, J.; Mendoza-Díaz, G. Chloro (histamine)(1, 10-Phenanthroline) Copper (II) Chloride Monohydrate. Acta Crystallogr. Sect. C Cryst. Struct. Commun. 2004, 60 (5), m205–m207. DOI: 10.1107/S0108270104006560
19. Melgar-Fernandez, R.; Demare, P.; Hong, E.; Rosas, M. A.; Escalante, J.; Munoz-Muniz, O.; Juaristi, E.; Regla, I.* Synthesis and Cardiovascular Activity of Metoprolol Analogues. Bioorg. Med. Chem. Lett. 2004, 14 (1), 191–194. DOI: 10.1016/j.bmcl.2003.09.070
18. Escalante, J.; Flores, P.; Priego, J. M. Synthesis of 2, 3-Dihydro-4 (1H)-Quinazollnones. Heterocycles-Sendai Inst. Heterocycl. Chem. 2004, 63 (9), 2019–2032. Online
17. Priego, J.; Flores, P.; Ortiz-Nava, C.; Escalante, J.* Synthesis of Enantiopure Cis-and Trans-2-Aminocyclohexane-1-Carboxylic Acids from Octahydroquinazolin-4-Ones. Tetrahedron: Asymmetry 2004, 15 (22), 3545–3549. DOI: 10.1016/j.tetasy.2004.08.032
16. Nicho, M. E.*; Hu, H.; López-Mata, C.; Escalante, J. Synthesis of Derivatives of Polythiophene and Their Application in an Electrochromic Device. Sol. Energy Mater. Sol. Cells 2004, 82 (1), 105–118. DOI: 10.1016/j.solmat.2004.01.009
2003
15. García‐Martínez, C.*; Cervantes‐Cuevas, H.; Escalante‐Garcia, J. Synthesis and NMR Configurational Analysis of 1, 3‐imidazolidin‐4‐ones Derived from (−)‐(S)‐phenylethylamine. Chirality 2003, 15 (S1), S74–S81. DOI: 10.1002/chir.10280
14. Escalante, J.*; González-Tototzin, M. A. Synthesis, Resolution and Absolute Configuration of Trans 4, 5-Diphenyl-Pyrrolidin-2-One: A Possible Chiral Auxiliary. Tetrahedron: Asymmetry 2003, 14 (8), 981–985. DOI: 10.1016/S0957-4166(03)00097-1
2002
13. Linzaga, I.; Escalante, J.; Muñoz, M.; Juaristi, E.* NMR and X-Ray Crystallographic Studies of Axial and Equatorial 2-Ethoxy-2-Oxo-1, 4, 2-Oxazaphosphinane. Tetrahedron 2002, 58 (44), 8973–8978. DOI: 10.1016/S0040-4020(02)01152-3
2001
12. Escalante, J.*; Hernández, A. L.; Juaristi, E.* Highly Diastereoselective Addition of a Racemic β-Alanine Enolate Derivative to Electrophiles. Rev. la Soc. 2001, 149 (4), 177–182. Online
11. Escalante, J.*; González-Tototzin, M. A.; Aviña, J.; Muñoz-Muñiz, O.; Juaristi, E*. Synthesis of β-Lactams and Cyclo-β-Dipeptides from β-Amino Acids: Experimental Observations and Theoretical Analysis. Tetrahedron 2001, 57 (10), 1883–1890. DOI: 10.1016/S0040-4020(00)01169-8
1999
10. Ramírez-Quirós, Y.; Balderas, M.; Escalante, J.; Quintana, D.; Gallardo, I.; Madrigal, D.; Molins, E.; Juaristi, E.* X-Ray Crystallographic Study of Substituted Perhydropyrimidinones. Extreme Changes in Ring Conformation. J. Org. Chem. 1999, 64 (23), 8668–8680. DOI: 10.1021/jo991297q
9. Juaristi, E.*; León-Romo, J. L.; Reyes, A.; Escalante, J. Recent Applications of α-Phenylethylamine (α-PEA) in the Preparation of Enantiopure Compounds. Part 3: α-PEA as Chiral Auxiliary. Part 4: α-PEA as Chiral Reagent in the Stereodifferentiation of Prochiral Substrates. Tetrahedron: Asymmetry 1999, 10 (13), 2441–2495. DOI: 10.1016/S0957-4166(99)00242-6
1998
8. Juaristi, E.*; López-Ruiz, H.; Madrigal, D.; Ramírez-Quirós, Y.; Escalante, J. α-Alkylation of (S)-Asparagine with Self-Regeneration of the Stereogenic Center: Enantioselective Synthesis of α-Substituted Aspartic Acids1, 2. J. Org. Chem. 1998, 63 (14), 4706–4710. DOI: 10.1021/jo980367a
7. Juaristi, E.*; Escalante, J.; León-Romo, J. L.; Reyes, A. Recent Applications of α-Phenylethylamine (α-PEA) in the Preparation of Enantiopure Compounds. Part 1: Incorporation in Chiral Catalysts. Part 2: α-PEA and Derivatives as Resolving Agents. Tetrahedron: Asymmetry 1998, 9 (5), 715–740. DOI: 10.1016/S0957-4166(98)00058-5
1997
6. Crich, D.*; Escalante, J.; Jiao, X.-Y. Solvent Effects in the β-(Phosphatoxy) Alkyl Radical Migration Asrevealed by Deuterium Labelling and 1H NMR Spectroscopy. J. Chem. Soc., Perkin Trans. 2 1997, No. 3, 627–630. DOI: 10.1039/A603916B
1995
5. Escalante, J.; Juaristi, E.* Enantioselective Synthesis of β-Amino Acids. 6. High 1, 2-Stereoinduction in the Preparation of Enantiopure 2 (R)-Hydroxy-3 (R)-N-Benzoylamino-3-Phenylpropionic Acid (like Stereoisomer of Taxol’s Side Chain). Tetrahedron Lett. 1995, 36 (25), 4397–4400. DOI: 10.1016/0040-4039(95)00859-B
1993
4. Juaristi, E.*; Escalante, J. Enantioselective Synthesis Of. Beta.-Amino Acids. 4. 1, 2 Asymmetric Induction in the Alkylation of 1-Benzoyl-3, 6 (S)-Dimethylperhydropyrimidin-4-One. Preparation of the like and Unlike Stereoisomers of 2-Methyl-and 2-Benzyl-3 (S)-Aminobutanoic Acid. J. Org. Chem. 1993, 58 (8), 2282–2285. DOI: 10.1021/jo00060a051
1992
3. Juaristi, E.*; Escalante, J.; Lamatsch, B.; Seebach, D. Enantioselective Synthesis Of. Beta.-Amino Acids. 2. Preparation of the like Stereoisomers of 2-Methyl-and 2-Benzyl-3-Aminobutanoic Acid. J. Org. Chem. 1992, 57 (8), 2396–2398. DOI: 10.1021/jo00034a037
2. Seebach, D.; Amatsch, B.; Amstutz, R.; Beck, A. K.; Doler, M.; Egli, M.; Fitzi, R.; Gautschi, M.; Herradön, B.; Hidber, P. C. Structure and Reactivity of Five‐and Six‐Ring N, N‐, N, O‐, and O, O‐acetals: A Lesson in Allylic 1, 3‐strain (A1, 3 Strain). Helv. Chim. Acta 1992, 75 (3), 913–934. DOI: 10.1002/hlca.19920750326
1991
1. Juaristi, E.*; Rizo, B.; Natal, V.; Escalante, J.; Regla, I. Alternative Method for the Resolution of 1-Benzoyl-2-Tert-Butyl-3-Methyl-1, 3-Imidazolidin-4-One. Tetrahedron: Asymmetry 1991, 2 (8), 821–826. DOI: 10.1016/S0957-4166(00)80465-6